SCHEMBL27800481

SCHEMBL27800481

CC(C)c1cccc(CCBr)n1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.37
NOS1 P29475 2/20 0.35
NOS2 P35228 2/20 0.35
ADORA2A P29274 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
CHRNA7 P36544 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4051420 0.84 CCR1 (0.40) KCNH2NOS1NOS2ADORA2ACHRNA7
SCHEMBL9974287 0.82 KCNH2 (0.47) KCNH2NOS1NOS2ADORA2A
SCHEMBL27778293 0.81 ADORA2A (0.36) KCNH2NOS1NOS2ADORA2ANPSR1
SCHEMBL12120627 0.81 SYK (0.40) KCNH2NOS1NOS2ADORA2A
SCHEMBL9232330 0.81 KCNH2 (0.37) KCNH2NOS1NOS2ADORA2ANPSR1
SCHEMBL8250521 0.79 KCNH2 (0.58) KCNH2NOS1NOS2ADORA2A
SCHEMBL20207664 0.78 CYP1A2 (0.36) KCNH2NOS1NOS2ADORA2ANPSR1
SCHEMBL1581851 0.78 KCNH2 (0.36) KCNH2NOS1NOS2ADORA2ACHRNA7
SCHEMBL27265753 0.78 SMN1; SMN2 (0.45) KCNH2NOS1NOS2NPSR1TDP1
SCHEMBL31481285 0.78 KCNH2 (0.36) KCNH2NOS1NOS2ADORA2ACHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101691370-A Triazolo[4,5-d] pyrimidine derivatives and their use as purinergic receptor antagonists VERNALIS RES LTD 2010-04-07 CN disclosed