SCHEMBL27802103

SCHEMBL27802103

COC(=O)c1cccc(CC(Br)Br)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 2/20 0.67
LOXL2 Q9Y4K0 1/20 0.64
CYP4F2 P78329 2/20 0.62
CYP4A11 Q02928 2/20 0.62
FOLH1 Q04609 1/20 0.58
HIF1A Q16665 1/20 0.52
MRGPRX4 Q96LA9 2/20 0.51
ALDH1A1 P00352 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
KDM4E B2RXH2 1/20 0.50
MAPT P10636 1/20 0.50
RAB9A P51151 1/20 0.50
HPGD P15428 1/20 0.48
TSHR P16473 1/20 0.47
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47
KMT2A Q03164 1/20 0.47
ABHD6 Q9BV23 1/20 0.46
HTT P42858 1/20 0.46
IDO1 P14902 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1790854 0.85 SLC7A5 (0.68) SLC7A5LOXL2CYP4F2CYP4A11FOLH1
SCHEMBL27781443 0.84 CYP4F2 (0.61) SLC7A5CYP4F2CYP4A11ALDH1A1SMN1; SMN2
SCHEMBL13589439 0.84 SLC7A5 (0.76) SLC7A5LOXL2CYP4F2CYP4A11FOLH1
SCHEMBL28281252 0.84 SLC7A5 (0.76) SLC7A5LOXL2CYP4F2CYP4A11FOLH1
SCHEMBL15609287 0.84 SLC7A5 (0.76) SLC7A5LOXL2CYP4F2CYP4A11FOLH1
SCHEMBL20168566 0.84 SLC7A5 (0.76) SLC7A5LOXL2CYP4F2CYP4A11FOLH1
SCHEMBL31276630 0.83 CYP4F2 (0.75) SLC7A5LOXL2CYP4F2CYP4A11FOLH1
SCHEMBL40012 0.83 CYP4F2 (0.75) SLC7A5LOXL2CYP4F2CYP4A11FOLH1
SCHEMBL27575558 0.83 SLC7A5 (0.58) SLC7A5LOXL2CYP4F2CYP4A11FOLH1
SCHEMBL6687519 0.83 SLC7A5 (0.69) SLC7A5LOXL2CYP4F2CYP4A11FOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101952254-B Isoquinoline modulators of ATP-binding cassette transporters VERTEX PHARMA 2012-09-05 CN disclosed
CN-101952254-A Isoquinoline modulators of ATP-binding cassette transporters VERTEX PHARMA 2011-01-19 CN disclosed