SCHEMBL27802465

SCHEMBL27802465

O=CC1CN(c2ncnc3[nH]nc(Br)c23)CCN1Cc1ccc(Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 13/20 0.42
RPS6KB1 P23443 2/20 0.37
KIT P10721 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL473344 0.86 AKT1 (0.41) AKT1RPS6KB1KITMEN1KMT2A
SCHEMBL473359 0.86 AKT1 (0.41) AKT1RPS6KB1KITMEN1KMT2A
SCHEMBL473424 0.85 AKT1 (0.42) AKT1RPS6KB1
SCHEMBL473311 0.81 MEN1 (0.50) AKT1RPS6KB1MEN1KMT2AALDH1A1
SCHEMBL473312 0.79 AKT1 (0.37) AKT1RPS6KB1MEN1KMT2A
SCHEMBL10159411 0.79 AKT1 (0.37) AKT1RPS6KB1KITMEN1KMT2A
SCHEMBL27802512 0.78 RPS6KB1 (0.41) AKT1RPS6KB1
SCHEMBL473308 0.77 AKT1 (0.46) AKT1RPS6KB1
SCHEMBL1790785 0.76 RPS6KB1 (0.47) AKT1RPS6KB1MEN1KMT2AALDH1A1
SCHEMBL473341 0.74 PDE10A (0.45) AKT1RPS6KB1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101959516-A Combination therapy comprising quinoxaline PI3K alpha inhibitors for the treatment of cancer EXELIXIS INC 2011-01-26 CN disclosed