SCHEMBL27802487

SCHEMBL27802487

NC(=O)N(Cc1cccc(-c2ccncc2)c1)c1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.46
MGLL Q99685 1/20 0.45
ABHD6 Q9BV23 2/20 0.41
STAT3 P40763 2/20 0.40
NR1H4 Q96RI1 1/20 0.40
BLM P54132 1/20 0.40
PRKCI P41743 1/20 0.40
CETP P11597 2/20 0.39
KDR P35968 1/20 0.39
GRM4 Q14833 1/20 0.39
PDK1 Q15118 1/20 0.39
MAPT P10636 1/20 0.39
BRAF P15056 2/20 0.38
CDK8 P49336 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4581453 0.92 S1PR1 (0.47) S1PR1MGLLABHD6STAT3NR1H4
SCHEMBL27802447 0.90 NR1H4 (0.47) S1PR1NR1H4CETPPDK1MAPT
SCHEMBL28786186 0.89 BLM (0.42) S1PR1BLMCETPKDRGRM4
SCHEMBL27802485 0.83 MKNK1 (0.46) S1PR1NR1H4KDRPDK1MAPT
SCHEMBL15104092 0.82 S1PR1 (0.41) S1PR1NR1H4KDRPDK1CDK8
SCHEMBL4583491 0.82 NR1H4 (0.48) S1PR1NR1H4CETPPDK1MAPT
SCHEMBL4582429 0.82 S1PR1 (0.46) S1PR1MGLLSTAT3NR1H4CETP
SCHEMBL4582467 0.82 BLM (0.44) S1PR1BLMCETPKDRGRM4
SCHEMBL1791462 0.78 BRAF (0.46) BLMKDRGRM4MAPTBRAF
SCHEMBL1790536 0.77 S1PR1 (0.44) S1PR1NR1H4CETPKDRGRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101959516-A Combination therapy comprising quinoxaline PI3K alpha inhibitors for the treatment of cancer EXELIXIS INC 2011-01-26 CN disclosed