SCHEMBL27808985

SCHEMBL27808985

CC(=O)Nc1cccc(CCc2ccc(CNC(=O)NN)cc2)n1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 6/20 0.47
PTPN1 P18031 1/20 0.45
NR3C2 P08235 1/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
MAPK8 P45983 1/20 0.41
MAOB P27338 1/20 0.38
ADORA2A P29274 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
MAP3K5 Q99683 1/20 0.37
PPID Q08752 1/20 0.37
EPHX1 P07099 1/20 0.37
MEN1 O00255 1/20 0.36
TP53 P04637 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27981485 0.99 AOC3 (0.47) AOC3PTPN1NR3C2KDM4ELMNA
SCHEMBL1432645 0.82 AOC3 (0.56) AOC3NR3C2KDM4ELMNASMN1; SMN2
SCHEMBL6788722 0.82 AOC3 (0.50) AOC3NR3C2KDM4ELMNANPSR1
Hydrochloric Acid SCHEMBL1432791 0.81 AOC3 (0.55) AOC3NR3C2KDM4ELMNASMN1; SMN2
SCHEMBL27808983 0.81 AOC3 (0.50) AOC3PTPN1NPC1PPID
Hydrochloric Acid SCHEMBL27981813 0.80 AOC3 (0.49) AOC3PTPN1NPC1PPID
SCHEMBL27808967 0.79 ACACB (0.43) PTPN1KDM4ELMNAMAPK8ADORA2A
SCHEMBL27808972 0.79 PTPN1 (0.66) AOC3PTPN1KDM4ELMNASMN1; SMN2
SCHEMBL973474 0.79 AOC3 (0.70) AOC3MAOBSMN1; SMN2KMT2A
Hydrochloric Acid SCHEMBL28813926 0.78 ACACB (0.42) PTPN1KDM4ELMNAMAPK8ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102046601-A Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R TECH UENO LTD 2011-05-04 CN claimed
CN-102046601-B Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R TECH UENO LTD 2014-08-27 CN disclosed
CN-102046601-A Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R TECH UENO LTD 2011-05-04 CN disclosed