SCHEMBL2780933

SCHEMBL2780933

OC[C@@]1(Cc2ccccc2)CNC[C@H]1c1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 9/20 0.49
RCOR1 Q9UKL0 5/20 0.49
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
MAOA P21397 6/20 0.36
MAOB P27338 6/20 0.36
ALDH1A1 P00352 1/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
REN P00797 2/20 0.34
CTSD P07339 1/20 0.34
CTSE P14091 1/20 0.34
PGC P20142 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11865200 0.93 KDM1A (0.40) KDM1ARCOR1SLC6A2SLC6A4SLC6A3
SCHEMBL11865318 0.90 KDM1A (0.44) KDM1ARCOR1MAOAMAOBALDH1A1
SCHEMBL1439673 0.90 KDM1A (0.47) KDM1ARCOR1MEN1KMT2AMAOA
Hydrochloric Acid SCHEMBL11860269 0.89 KDM1A (0.45) KDM1ARCOR1MAOAMAOBALDH1A1
SCHEMBL2225021 0.87 KDM1A (0.52) KDM1ARCOR1MAOAMAOBSLC6A2
SCHEMBL1421527 0.87 KDM1A (0.52) KDM1ARCOR1MAOAMAOBSLC6A2
SCHEMBL2784188 0.86 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3
SCHEMBL1439732 0.84 KDM1A (0.46) KDM1ARCOR1MAOAMAOBSLC6A2
SCHEMBL3715321 0.80 KDM1A (0.45) KDM1ARCOR1MEN1KMT2AMAOA
SCHEMBL3712746 0.80 KDM1A (0.45) KDM1ARCOR1MEN1KMT2AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2398768-A1 PYRROLIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2011-12-28 EP disclosed
WO-2010094667-A1 PYRROLIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-08-26 WO disclosed