SCHEMBL27853041

SCHEMBL27853041

O=C(O)CC1CCNC(c2cccc(C(F)(F)F)c2)C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.45
KDM1A O60341 2/20 0.43
FFAR1 O14842 2/20 0.43
DGAT1 O75907 1/20 0.41
SOAT1 P35610 1/20 0.41
FFAR4 Q5NUL3 4/20 0.40
S1PR4 O95977 1/20 0.40
S1PR1 P21453 1/20 0.40
S1PR3 Q99500 1/20 0.40
S1PR5 Q9H228 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2B P41595 1/20 0.40
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HTT P42858 1/20 0.39
HTR1A P08908 1/20 0.38
USP5 P45974 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2860924 0.99 HTR2C (0.46) HTR2CKDM1AFFAR1DGAT1SOAT1
SCHEMBL27869978 0.88 FFAR1 (0.37) FFAR1FFAR4S1PR4S1PR1S1PR3
SCHEMBL13604396 0.86 GUSB (0.43) HTR2CKDM1ALMNAMAPTSMN1; SMN2
SCHEMBL2493402 0.85 PSEN1 (0.45) HTR2CKDM1ADGAT1SOAT1FFAR4
SCHEMBL21820688 0.85 PSEN1 (0.45) HTR2CKDM1ADGAT1SOAT1FFAR4
SCHEMBL4493249 0.85 PSEN1 (0.45) HTR2CKDM1ADGAT1SOAT1FFAR4
SCHEMBL2861143 0.85 PSEN1 (0.45) HTR2CKDM1ADGAT1SOAT1FFAR4
Hydrochloric Acid SCHEMBL2874986 0.84 PSEN1 (0.44) HTR2CKDM1ADGAT1SOAT1FFAR4
Hydrochloric Acid SCHEMBL2161847 0.84 PSEN1 (0.44) HTR2CKDM1ADGAT1SOAT1FFAR4
SCHEMBL2852835 0.82 FFAR4 (0.47) KDM1ADGAT1SOAT1FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102459246-B Isoxazol-3 (2H) -one analogs as therapeutic agents ASTRAZENECA AB 2014-05-07 CN disclosed
CN-102459246-A Isoxazol-3 (2H) -one analogs as therapeutic agents ASTRAZENECA AB 2012-05-16 CN disclosed