SCHEMBL27856466

SCHEMBL27856466

Cc1nn(-c2cnc(C#N)c(NCCc3ccccn3)c2)c2cccc(-c3cnc4ccccc4c3)c12

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 15/20 0.50
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36
KCNA5 P22460 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL426294 0.86 HSP90AA1 (0.60) HSP90AA1
SCHEMBL2184084 0.85 HSP90AA1 (0.45) HSP90AA1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL421919 0.85 HSP90AA1 (0.44) HSP90AA1SMN1; SMN2
SCHEMBL27856465 0.85 HSP90AA1 (0.45) HSP90AA1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL1394276 0.85 HSP90AA1 (0.51) HSP90AA1
SCHEMBL1395213 0.79 HSP90AA1 (0.59) HSP90AA1
SCHEMBL1395132 0.79 HSP90AA1 (0.71) HSP90AA1
SCHEMBL1395131 0.79 HSP90AA1 (0.71) HSP90AA1
SCHEMBL1394528 0.78 HSP90AA1 (0.52) HSP90AA1
SCHEMBL460350 0.77 HSP90AA1 (0.48) HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102439003-A Indazole derivatives inhibiting HSP90, compositions containing said derivatives and uses thereof SANOFI AVENTIS 2012-05-02 CN disclosed