SCHEMBL27859244

SCHEMBL27859244

c1ncc(-n2cncn2)cn1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.61
KDM4E B2RXH2 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 1/20 0.50
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
FBP1 P09467 1/20 0.40
LMNA P02545 1/20 0.34
HSP90AA1 P07900 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
DPP4 P27487 2/20 0.33
CYP11B2 P19099 1/20 0.33
BRS3 P32247 1/20 0.33
MAPK10 P53779 1/20 0.33
HTR1A P08908 1/20 0.32
HTR2C P28335 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27905069 0.79 SMN1; SMN2 (0.72) CYP2A6KDM4ESMN1; SMN2ALDH1A1CYP1A2
SCHEMBL2730703 0.76 CYP2A6 (1.00) CYP2A6KDM4ESMN1; SMN2ALDH1A1CYP1A2
SCHEMBL9363173 0.75 KDM4E (0.60) CYP2A6KDM4ESMN1; SMN2ALDH1A1CYP1A2
SCHEMBL25614362 0.74 CYP2A6 (0.50) CYP2A6KDM4ESMN1; SMN2ALDH1A1CYP1A2
SCHEMBL31157148 0.74 CYP2A6 (0.50) CYP2A6KDM4ESMN1; SMN2ALDH1A1CYP1A2
SCHEMBL3315428 0.74 CYP2A6 (0.50) CYP2A6KDM4ESMN1; SMN2ALDH1A1CYP1A2
SCHEMBL1009561 0.73 CYP2A6 (0.64) CYP2A6KDM4ESMN1; SMN2ALDH1A1CYP1A2
SCHEMBL10508046 0.73 SMN1; SMN2 (0.59) CYP2A6KDM4ESMN1; SMN2ALDH1A1CYP1A2
SCHEMBL28108762 0.73 KDM4E (0.64) CYP2A6KDM4ESMN1; SMN2ALDH1A1CYP1A2
SCHEMBL12414654 0.73 CYP2A6 (0.44) CYP2A6KDM4ESMN1; SMN2ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105008346-B Pyrimidine derivatives as phosphodiesterase 10(PDE-10) inhibitors 帕罗生物制药有限公司 2018-11-13 CN disclosed
CN-102548980-A 5-fluoropyrimidinone derivatives DOW AGROSCIENCES LLC 2012-07-04 CN disclosed