SCHEMBL27859971

SCHEMBL27859971

O=C(O)[C@H]1CCCN(CC(O)c2ccc(-c3noc(-c4cnn(-c5ccccn5)c4C(F)(F)F)n3)cc2)C1

nearest known ligand 0.66

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.66
S1PR3 Q99500 15/20 0.62
S1PR4 O95977 2/20 0.62
S1PR5 Q9H228 2/20 0.62
CYP2C8 P10632 1/20 0.51
KCNH2 Q12809 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1226622 1.00 S1PR1 (0.66) S1PR1S1PR3S1PR4S1PR5CYP2C8
SCHEMBL1226619 1.00 S1PR1 (0.66) S1PR1S1PR3S1PR4S1PR5CYP2C8
SCHEMBL1226614 1.00 S1PR1 (0.66) S1PR1S1PR3S1PR4S1PR5CYP2C8
SCHEMBL1227287 0.91 S1PR1 (0.66) S1PR1S1PR3S1PR4S1PR5CYP2C8
SCHEMBL1227279 0.91 S1PR1 (0.66) S1PR1S1PR3S1PR4S1PR5CYP2C8
SCHEMBL1227283 0.91 S1PR1 (0.66) S1PR1S1PR3S1PR4S1PR5CYP2C8
SCHEMBL27876340 0.91 S1PR1 (0.66) S1PR1S1PR3S1PR4S1PR5CYP2C8
SCHEMBL1225710 0.91 S1PR1 (0.67) S1PR1S1PR3S1PR4S1PR5CYP2C8
SCHEMBL1225704 0.91 S1PR1 (0.67) S1PR1S1PR3S1PR4S1PR5CYP2C8
SCHEMBL1225701 0.91 S1PR1 (0.67) S1PR1S1PR3S1PR4S1PR5CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102548989-A Sphingosine-1-phosphate receptor agonists BRISTOL MYERS SQUIBB CO 2012-07-04 CN claimed
CN-102548989-A Sphingosine-1-phosphate receptor agonists BRISTOL MYERS SQUIBB CO 2012-07-04 CN disclosed