SCHEMBL27870871

SCHEMBL27870871

Cc1ccc(-c2ccccn2)c(C(=O)c2cc(C)ccc2-c2ccccn2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.48
HCRTR1 O43613 12/20 0.47
TUBB4A P04350 1/20 0.46
TUBB P07437 1/20 0.46
TUBA3C P0DPH7 1/20 0.46
TUBA1B P68363 1/20 0.46
TUBA4A P68366 1/20 0.46
TUBB4B P68371 1/20 0.46
TUBB3 Q13509 1/20 0.46
TUBB2A Q13885 1/20 0.46
TUBB8 Q3ZCM7 1/20 0.46
TUBA3E Q6PEY2 1/20 0.46
TUBA1A Q71U36 1/20 0.46
TUBA1C Q9BQE3 1/20 0.46
TUBB6 Q9BUF5 1/20 0.46
TUBB2B Q9BVA1 1/20 0.46
TUBB1 Q9H4B7 1/20 0.46
HCRTR2 O43614 8/20 0.45
BRD4 O60885 1/20 0.44
BRD2 P25440 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9955206 0.89 KDM4E (0.47) BTKHCRTR1BRD4BRD2BRD3
SCHEMBL29814525 0.89 KDM4E (0.47) BTKHCRTR1BRD4BRD2BRD3
SCHEMBL19499711 0.89 BRD4 (0.50) BTKHCRTR1TUBB4ATUBBTUBA3C
SCHEMBL9955328 0.85 CYP46A1 (0.63) BTKHCRTR1TUBB4ATUBBTUBA3C
SCHEMBL27870875 0.81 HCRTR1 (0.54) HCRTR1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL5330963 0.80 NPC1 (0.49) BTKBRD4BRD2BRD3BAZ2B
SCHEMBL22468515 0.79 KDM4E (0.47) BTKBRD4BRD2BRD3BAZ2B
SCHEMBL27870880 0.79 CYP46A1 (0.46) HCRTR1HCRTR2KDM4ENPC1RAB9A
SCHEMBL3423163 0.79 KDM4E (0.50) BTKKDM4ENPC1ALDH1A1TP53
SCHEMBL9202323 0.79 KDM4E (0.50) HCRTR1HCRTR2BRD4BRD2BRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102471314-A Spiro amino compounds suitable for the treatment of inter alia sleep disorders and drug addiction ROTTAPHARM SPA 2012-05-23 CN disclosed