SCHEMBL27870993

SCHEMBL27870993

CC(c1nc(-c2ccc(-c3ccc4cc(-c5c[nH]c(C(C)N(C)C(=O)OC(C)(C)C)n5)ccc4c3)cc2)c[nH]1)N(C)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 4/20 0.40
PAX8 Q06710 1/20 0.34
FFAR4 Q5NUL3 1/20 0.33
GSK3B P49841 1/20 0.32
DYRK1A Q13627 1/20 0.32
MCL1 Q07820 1/20 0.31
SGK1 O00141 1/20 0.31
ALPL P05186 1/20 0.31
PDGFRB P09619 1/20 0.30
SCN9A Q15858 1/20 0.30
TTK P33981 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27870991 1.00 AAK1 (0.40) AAK1PAX8FFAR4GSK3BDYRK1A
SCHEMBL1294210 0.96 AAK1 (0.38) AAK1PAX8FFAR4GSK3BDYRK1A
SCHEMBL27887125 0.92 AAK1 (0.36) AAK1PAX8GSK3BDYRK1A
SCHEMBL19690733 0.91 AAK1 (0.35) AAK1GSK3BDYRK1A
SCHEMBL1293882 0.90 AAK1 (0.36) AAK1FFAR4
SCHEMBL1294208 0.89 AAK1 (0.36) AAK1FFAR4SCN9A
SCHEMBL1293881 0.88 AAK1 (0.35) AAK1FFAR4
SCHEMBL1293879 0.88 AAK1 (0.34) AAK1GSK3BDYRK1ASCN9A
SCHEMBL9980531 0.88 AAK1 (0.36) AAK1PAX8
SCHEMBL10182576 0.88 AAK1 (0.37) AAK1PAX8MCL1ALPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102712623-B Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2014-04-02 CN disclosed
CN-102712623-A Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2012-10-03 CN disclosed
CN-102686565-A Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2012-09-19 CN disclosed