Benzothiophene

Benzothiophene

SCHEMBL27872206

O=Cc1ccccc1.c1ccc2sccc2c1

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.56
ALDH1A1 P00352 3/20 0.54
CTNNB1 P35222 1/20 0.38
WNT3A P56704 1/20 0.38
CA12 O43570 2/20 0.35
CA9 Q16790 1/20 0.35
KMT2A Q03164 2/20 0.34
CA2 P00918 1/20 0.34
CSNK2A2 P19784 1/20 0.33
CSNK2B P67870 1/20 0.33
CSNK2A1 P68400 1/20 0.33
PTGS1 P23219 1/20 0.33
PPARG P37231 1/20 0.33
TRPA1 O75762 1/20 0.33
LMNA P02545 1/20 0.33
ALOX5 P09917 1/20 0.33
MAPK1 P28482 1/20 0.33
MEN1 O00255 1/20 0.33
RAB9A P51151 1/20 0.33
PTPRC P08575 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzothiophene SCHEMBL15227137 0.83 CTNNB1 (0.43) CYP2A6CTNNB1WNT3ACA12CA9
Benzothiophene SCHEMBL28493798 0.83 CYP2A6 (0.51) CYP2A6ALDH1A1CTNNB1WNT3ACA12
Benzothiophene SCHEMBL28112179 0.82 CYP2A6 (0.47) CYP2A6CTNNB1WNT3ACA12CA9
Benzothiophene SCHEMBL30395947 0.82 CYP2A6 (0.47) CYP2A6CTNNB1WNT3ACA12CA9
Benzothiophene SCHEMBL28030266 0.82 CYP2A6 (0.47) CYP2A6CTNNB1WNT3ACA12CA9
Benzothiophene SCHEMBL28882160 0.82 CYP2A6 (0.47) CYP2A6CTNNB1WNT3ACA12CA9
Benzothiophene SCHEMBL28758675 0.81 CTNNB1 (0.46) CYP2A6CTNNB1WNT3ACA12CA9
Benzothiophene SCHEMBL4378682 0.81 CTNNB1 (0.46) CYP2A6CTNNB1WNT3ACA12CA9
Benzothiophene SCHEMBL7023 0.81
Benzothiophene SCHEMBL253491 0.81 CA12 (0.42) CYP2A6ALDH1A1CTNNB1WNT3ACA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102690256-B Phenyl benzothiophene ketone compound and preparation method and application thereof UNIV SHANXI 2013-09-04 CN claimed
CN-102690256-A Phenyl benzothiophene ketone compound and preparation method and application thereof UNIV SHANXI 2012-09-26 CN claimed
CN-102690256-B Phenyl benzothiophene ketone compound and preparation method and application thereof UNIV SHANXI 2013-09-04 CN disclosed
CN-102690256-B Phenyl benzothiophene ketone compound and preparation method and application thereof UNIV SHANXI 2013-09-04 CN disclosed
CN-102690256-B Phenyl benzothiophene ketone compound and preparation method and application thereof UNIV SHANXI 2013-09-04 CN disclosed
CN-102690256-A Phenyl benzothiophene ketone compound and preparation method and application thereof UNIV SHANXI 2012-09-26 CN disclosed
CN-102690256-A Phenyl benzothiophene ketone compound and preparation method and application thereof UNIV SHANXI 2012-09-26 CN disclosed
CN-102690256-A Phenyl benzothiophene ketone compound and preparation method and application thereof UNIV SHANXI 2012-09-26 CN disclosed