SCHEMBL27878418

SCHEMBL27878418

CCCOc1c(C)cc(-c2nnc(-c3cc(C)c(CC(C)C)s3)o2)cc1CC

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 19/20 0.41
S1PR3 Q99500 15/20 0.41
S1PR5 Q9H228 1/20 0.39
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL263225 0.86 S1PR1 (0.50) S1PR1S1PR3S1PR5
SCHEMBL262084 0.86 S1PR1 (0.50) S1PR1S1PR3S1PR5
SCHEMBL263803 0.82 S1PR1 (0.34) S1PR1S1PR3S1PR5
SCHEMBL262105 0.80 S1PR1 (0.66) S1PR1S1PR3S1PR5
SCHEMBL262404 0.80 S1PR1 (0.66) S1PR1S1PR3S1PR5
SCHEMBL27869684 0.72 S1PR1 (0.40) S1PR1S1PR3KDM4ENPC1ALDH1A1
SCHEMBL27869697 0.70 S1PR1 (0.42) S1PR1S1PR3KDM4ENPC1ALDH1A1
SCHEMBL14285688 0.70 S1PR1 (0.43) S1PR1S1PR3KDM4ENPC1ALDH1A1
SCHEMBL2294514 0.69 S1PR1 (0.70) S1PR1S1PR3
SCHEMBL2291664 0.69 S1PR1 (0.70) S1PR1S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101528726-B Thiophene derivatives as S1P1/EDG1 receptor agonists ACTELION PHARMACEUTICALS LTD 2012-11-14 CN disclosed