SCHEMBL2788461

SCHEMBL2788461

CN(C)CCN(C(=O)O)c1cccc2[nH]cnc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.44
ALDH1A1 P00352 2/20 0.41
PKM P14618 1/20 0.41
EGLN1 Q9GZT9 1/20 0.39
KDM4E B2RXH2 1/20 0.36
HTR2C P28335 2/20 0.36
KDM4A O75164 1/20 0.35
KDM4B O94953 1/20 0.35
KDM5C P41229 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTR1A P08908 1/20 0.34
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
MAOA P21397 1/20 0.34
ADRA1D P25100 1/20 0.34
HTR1B P28222 1/20 0.34
HTR2A P28223 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7032511 0.78 PARP1 (0.47) PARP1ALDH1A1PKM
SCHEMBL7031817 0.75 PARP1 (0.43) PARP1ALDH1A1KDM4E
SCHEMBL31693421 0.71 HTR2A (0.47) PARP1ALDH1A1PKMHTR2CHTR1A
SCHEMBL29907275 0.70 PARP1 (0.43) PARP1ALDH1A1PKM
SCHEMBL27146952 0.70 PARP1 (0.43) PARP1ALDH1A1PKM
SCHEMBL29337474 0.69 PARP1 (0.40) PARP1ALDH1A1PKM
SCHEMBL29907247 0.69 BRD4 (0.42) PARP1ALDH1A1PKMHTR2CHTR1A
SCHEMBL27143088 0.69 BRD4 (0.42) PARP1ALDH1A1PKMHTR2CHTR1A
SCHEMBL27644639 0.69 PARP1 (0.43) PARP1CYP2C19
SCHEMBL2128520 0.68 PARP1 (0.64) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010110686-A1 PYRIMIDINYL AND 1,3,5 TRIAZINYL BENZIMIDAZOLES AND THEIR USE IN CANCER THERAPY PATHWAY THERAPEUTICS LIMITED (NZ) 2010-09-30 WO disclosed