SCHEMBL27887643

SCHEMBL27887643

CO[C@H]1CCCN1c1nc(-n2cccn2)nc(N)c1Br

nearest known ligand 0.76

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 18/20 0.76
ADORA3 P0DMS8 1/20 0.57
ADORA2B P29275 1/20 0.57
ADORA1 P30542 1/20 0.57
PDE10A Q9Y233 1/20 0.41
ADK P55263 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27904499 1.00 ADORA2A (0.76) ADORA2AADORA3ADORA2BADORA1PDE10A
SCHEMBL27887645 1.00 ADORA2A (0.76) ADORA2AADORA3ADORA2BADORA1PDE10A
SCHEMBL2555841 0.86 ADORA2A (1.00) ADORA2AADORA3ADORA2BADORA1PDE10A
SCHEMBL2555844 0.86 ADORA2A (1.00) ADORA2AADORA3ADORA2BADORA1PDE10A
SCHEMBL2542194 0.85 ADORA2A (0.70) ADORA2AADORA3ADORA2BADORA1PDE10A
SCHEMBL2548740 0.85 ADORA2A (0.70) ADORA2AADORA3ADORA2BADORA1PDE10A
SCHEMBL2555110 0.80 ADORA2A (0.76) ADORA2AADORA3ADORA2BADORA1PDE10A
SCHEMBL2555106 0.80 ADORA2A (0.76) ADORA2AADORA3ADORA2BADORA1PDE10A
SCHEMBL2556664 0.80 ADORA2A (0.76) ADORA2AADORA3ADORA2BADORA1PDE10A
SCHEMBL2550783 0.76 ADORA2A (0.79) ADORA2AADORA3ADORA2BADORA1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102892761-A 4 - aminopyrimidine derivatives and their as as adenosine a2a receptor antagonists PALOBIOFARMA SL 2013-01-23 CN disclosed