SCHEMBL27896017

SCHEMBL27896017

CC(C)c1nnn(-c2c(Cl)cccc2Cl)c1CCBr

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.43
GABRB3 P28472 10/20 0.33
GABRA2 P47869 3/20 0.32
GABRB2 P47870 3/20 0.32
CCNK O75909 1/20 0.31
CCND3 P30281 1/20 0.31
GSK3B P49841 1/20 0.31
CDK7 P50613 1/20 0.31
CDK9 P50750 1/20 0.31
CCNH P51946 1/20 0.31
CDK6 Q00534 1/20 0.31
CDK12 Q9NYV4 1/20 0.31
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1096680 0.89 NR1H4 (0.45) NR1H4GABRB3GABRA2GABRB2CCNK
SCHEMBL498069 0.87 NR1H4 (0.45) NR1H4GABRB3GABRA2GABRB2CCNK
SCHEMBL12188553 0.84 NR1H4 (0.45) NR1H4GABRB3GABRA2GABRB2CCNK
SCHEMBL498227 0.83 NR1H4 (0.47) NR1H4GABRB3GABRA2GABRB2CCNK
SCHEMBL12878994 0.76 NR1H4 (0.39) NR1H4GABRB3GABRA2GABRB2CCNK
SCHEMBL498141 0.76 NR1H4 (0.49) NR1H4CCNKCCND3GSK3BCDK7
SCHEMBL27896299 0.75 NR1H4 (0.43) NR1H4RORC
SCHEMBL498805 0.74 NR1H4 (0.56) NR1H4CCNKCCND3GSK3BCDK7
SCHEMBL27896015 0.72 NR1H4 (0.39) NR1H4CCNKCCND3GSK3BCDK7
SCHEMBL12168764 0.72 NR1H4 (0.37) NR1H4CCNKCCND3GSK3BCDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101743232-B Compounds and methods for modulating fxr LILLY CO ELI 2013-03-06 CN disclosed