SCHEMBL2790219

SCHEMBL2790219

COCCCn1c(C2CCCN(C(=O)C[C@@H](Cc3ccc(-c4ccc(C(=O)O)cc4)cc3)NC(=O)OC(C)(C)C)C2)cc2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PADI4 Q9UM07 3/20 0.41
KLK5 Q9Y337 1/20 0.39
HRH2 P25021 1/20 0.38
HRH1 P35367 1/20 0.38
PROKR1 Q8TCW9 5/20 0.37
CNR2 P34972 2/20 0.37
PTGER4 P35408 2/20 0.36
ACE P12821 1/20 0.35
CMA1 P23946 1/20 0.34
USP30 Q70CQ3 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7897490 0.92 PADI4 (0.41) PADI4KLK5HRH2HRH1PROKR1
SCHEMBL7891183 0.91 PADI4 (0.40) PADI4KLK5HRH2HRH1PROKR1
SCHEMBL739547 0.88 HRH1 (0.41) PADI4KLK5HRH2HRH1PTGER4
SCHEMBL739548 0.88 HRH1 (0.41) PADI4KLK5HRH2HRH1PTGER4
SCHEMBL7897738 0.86 PADI4 (0.37) PADI4KLK5HRH2HRH1PROKR1
SCHEMBL2791389 0.85 CNR2 (0.40) PADI4PROKR1CNR2PTGER4
SCHEMBL763858 0.84 KCNH2 (0.42) KLK5HRH2HRH1ACE
SCHEMBL739119 0.83 HRH1 (0.39) HRH2HRH1
SCHEMBL739120 0.83 HRH1 (0.39) HRH2HRH1
SCHEMBL2791612 0.83 PROKR1 (0.39) PADI4PROKR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed