SCHEMBL2790784

SCHEMBL2790784

N#Cc1[nH]c2ccc(C3(Cc4ccccc4)CCNC3)cc2c1C(F)(F)C(=O)OF

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 18/20 0.54
SLC6A4 P31645 18/20 0.54
SLC6A3 Q01959 18/20 0.54
CYP2D6 P10635 16/20 0.54
KCNH2 Q12809 5/20 0.53
TACR1 P25103 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL980900 0.84 SLC6A2 (0.55) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL2777923 0.79 SLC6A2 (0.55) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
Trifluoroacetic Acid SCHEMBL980899 0.74 SLC6A2 (0.83) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL986649 0.71 SLC6A4 (1.00) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL982193 0.70 SLC6A2 (0.51) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL984751 0.70 SLC6A2 (0.76) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL980786 0.70 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL984544 0.67 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL982643 0.66 SLC6A2 (0.82) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
Hydrochloric Acid SCHEMBL984497 0.66 SLC6A2 (0.81) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257545-A1 PYRROLIDINYL DERIVATIVES AND USES THEREOF F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009115427-A1 PYRROLIDINYL DERIVATIVES AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2009-09-24 WO disclosed