SCHEMBL27923769

SCHEMBL27923769

Cc1cc(C)cc(CC(c2cccc(F)c2)c2nc(-c3ccc(CN4CC(C(=O)O)C4)cc3)no2)c1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.54
S1PR5 Q9H228 11/20 0.54
S1PR4 O95977 9/20 0.54
S1PR3 Q99500 9/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27942795 0.93 S1PR1 (0.56) S1PR1S1PR5S1PR4S1PR3
SCHEMBL9107811 0.91 S1PR1 (0.53) S1PR1S1PR5S1PR4S1PR3
SCHEMBL27942984 0.91 S1PR1 (0.54) S1PR1S1PR5S1PR4S1PR3
SCHEMBL28808364 0.90 S1PR1 (0.60) S1PR1S1PR5S1PR4S1PR3
SCHEMBL27923772 0.90 S1PR5 (0.54) S1PR1S1PR5S1PR4S1PR3
SCHEMBL27942799 0.85 S1PR1 (0.54) S1PR1S1PR5S1PR4S1PR3
SCHEMBL27923768 0.85 S1PR1 (0.54) S1PR1S1PR5S1PR4S1PR3
SCHEMBL9105697 0.84 S1PR1 (0.55) S1PR1S1PR5S1PR4S1PR3
SCHEMBL9106954 0.83 S1PR1 (0.57) S1PR1S1PR5S1PR4S1PR3
SCHEMBL27923774 0.83 S1PR1 (0.54) S1PR1S1PR5S1PR4S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103370065-A Novel benzyl azetidine derivatives as sphingosine 1-phosphate (S1P) receptor modulators ALLERGAN INC 2013-10-23 CN claimed
CN-103370065-A Novel benzyl azetidine derivatives as sphingosine 1-phosphate (S1P) receptor modulators ALLERGAN INC 2013-10-23 CN disclosed