SCHEMBL27940964

SCHEMBL27940964

COc1cccc(-c2ccnc(Nc3cccc([N+](=O)[O-])c3)c2)c1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 10/20 0.59
ROCK1 Q13464 1/20 0.53
AKR1C3 P42330 1/20 0.51
AKR1C2 P52895 1/20 0.51
ABL1 P00519 2/20 0.49
BCR P11274 2/20 0.49
PRKCA P17252 2/20 0.49
ABCC1 P33527 1/20 0.49
EGFR P00533 3/20 0.48
SRC P12931 1/20 0.48
PTGES O14684 1/20 0.47
ALOX5 P09917 1/20 0.47
TNNI3K Q59H18 1/20 0.47
MEN1 O00255 1/20 0.47
MAPT P10636 1/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12487318 0.82 ABCG2 (0.56) ABCG2ROCK1ABL1BCRPRKCA
SCHEMBL27112560 0.81 MEN1 (0.55) ABCG2ROCK1ABCC1EGFRMEN1
SCHEMBL4736155 0.81 ABL1 (0.71) ABCG2ABL1BCRPRKCAEGFR
SCHEMBL14254280 0.81 EGFR (0.50) ABCG2ROCK1EGFRMEN1MAPT
SCHEMBL5468622 0.80 AKR1C3 (0.64) ABCG2AKR1C3AKR1C2PTGESALOX5
SCHEMBL12486792 0.79 ABCG2 (0.50) ABCG2ROCK1AKR1C3AKR1C2ABL1
SCHEMBL30469306 0.78 MAOB (0.60) ABCG2MEN1MAPTMAPK1HTT
SCHEMBL20557970 0.78 MAOB (0.60) ABCG2MEN1MAPTMAPK1HTT
SCHEMBL27940856 0.78 TNNI3K (0.56) ROCK1ABL1EGFRTNNI3KMEN1
SCHEMBL28807899 0.77 EGFR (0.60) ROCK1EGFRTNNI3K

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103562184-A Pharmaceutically active disubstituted pyridine derivatives LEAD DISCOVERY CENTER GMBH 2014-02-05 CN claimed