SCHEMBL27960992

SCHEMBL27960992

COC(=O)CCC1(N)CCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.46
LMNA P02545 4/20 0.39
KDM4E B2RXH2 1/20 0.39
KMT2A Q03164 3/20 0.36
MEN1 O00255 1/20 0.36
CA12 O43570 1/20 0.35
CA14 Q9ULX7 1/20 0.35
HSD17B10 Q99714 2/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
EPHX2 P34913 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MGAM O43451 1/20 0.33
GAA P10253 1/20 0.33
SI P14410 1/20 0.33
MGAM2 Q2M2H8 1/20 0.33
SLC1A1 P43005 1/20 0.33
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29087328 0.96 TSHR (0.46) TSHRLMNAKDM4EKMT2AMEN1
SCHEMBL3447711 0.94 TSHR (0.44) TSHRLMNAKDM4EKMT2AMEN1
SCHEMBL14151827 0.92 TSHR (0.50) TSHRLMNAKDM4EKMT2AMEN1
SCHEMBL18402675 0.83 TSHR (0.48) TSHRLMNAKDM4EKMT2AMEN1
SCHEMBL28207119 0.83 TSHR (0.48) TSHRLMNAKDM4EKMT2AALDH1A1
SCHEMBL27623828 0.80 TSHR (0.54) TSHRLMNAKDM4EKMT2AMEN1
SCHEMBL23890366 0.79 TSHR (0.41) TSHRLMNAKDM4EKMT2AMEN1
SCHEMBL15621351 0.79 TSHR (0.39) TSHRLMNAKDM4EHSD17B10ALDH1A1
SCHEMBL8252653 0.78 TSHR (0.48) TSHRLMNAKDM4EKMT2AMEN1
SCHEMBL15539095 0.77 TSHR (0.52) TSHRLMNAKDM4EKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105503862-B Inhibitors of influenza viruses replication 沃泰克斯药物股份有限公司 2018-02-02 CN disclosed
CN-105503862-A Inhibitors of influenza virus replication VERTEX PHARMA 2016-04-20 CN disclosed
CN-105481853-A Inhibitors of influenza viruses replication VERTEX PHARMA 2016-04-13 CN disclosed
CN-103764654-B Inhibitors of influenza virus replication VERTEX PHARMACEUTICALS INC. (US) 2016-01-20 CN disclosed
CN-103764654-A Inhibitors of influenza virus replication VERTEX PHARMA 2014-04-30 CN disclosed