SCHEMBL27976752

SCHEMBL27976752

COc1ccc(-c2ccc3cncnc3c2)cc1

nearest known ligand 0.76

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.76
PDGFRB P09619 2/20 0.51
PDGFRA P16234 2/20 0.51
MAP4K4 O95819 1/20 0.50
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
CYP11B1 P15538 3/20 0.48
CYP11B2 P19099 3/20 0.48
CASP3 P42574 1/20 0.47
SENP7 Q9BQF6 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
KMT2A Q03164 1/20 0.47
DYRK1A Q13627 2/20 0.46
FGFR4 P22455 1/20 0.46
CYP17A1 P05093 1/20 0.45
CYP19A1 P11511 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28158032 0.87 EGFR (0.76) EGFRPDGFRBPDGFRAMAP4K4CYP11B1
SCHEMBL668493 0.86 EGFR (1.00) EGFRPDGFRBPDGFRANPC1RAB9A
SCHEMBL30241125 0.86 EGFR (1.00) EGFRPDGFRBPDGFRANPC1RAB9A
SCHEMBL29517021 0.86 EGFR (1.00) EGFRPDGFRBPDGFRANPC1RAB9A
Hydrochloric Acid SCHEMBL28023744 0.85 EGFR (0.96) EGFRPDGFRBPDGFRANPC1RAB9A
SCHEMBL8641138 0.84 EGFR (0.64) EGFRFGFR4
SCHEMBL27991038 0.81 EGFR (0.53) EGFRPDGFRBPDGFRAFGFR4
SCHEMBL21982453 0.80 EGFR (0.57) EGFRMAP4K4NPC1CYP11B1CYP11B2
SCHEMBL28127970 0.79 EGFR (0.68) EGFRPDGFRBPDGFRANPC1RAB9A
SCHEMBL28127969 0.79 EGFR (0.68) EGFRPDGFRBPDGFRANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102675222-B Method for preparing multi-substituted quinazoline and heterocyclic pyrimidine derivative UNIV TSINGHUA 2014-11-26 CN disclosed
CN-102675223-B Preparation method for polysubstitution quinazoline and heterocyclic ring pyrimidine derivative UNIV TSINGHUA 2014-08-27 CN disclosed