SCHEMBL27979210

SCHEMBL27979210

O=C(CCc1ccc(Br)c(F)c1)CCc1ccc(Br)c(F)c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IAPP P10997 3/20 0.45
FFAR4 Q5NUL3 3/20 0.42
FFAR1 O14842 2/20 0.42
ALOX5 P09917 1/20 0.38
OR51E2 Q9H255 1/20 0.38
KIF11 P52732 1/20 0.38
PTPRB P23467 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C8 P10632 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2B6 P20813 1/20 0.36
CYP2C19 P33261 1/20 0.36
F2RL1 P55085 1/20 0.36
SLC5A1 P13866 1/20 0.36
SLC5A2 P31639 1/20 0.36
POLB P06746 1/20 0.36
RAB9A P51151 1/20 0.36
CCR5 P51681 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30816271 0.87 FFAR1 (0.55) FFAR4FFAR1PTPRB
SCHEMBL9247568 0.87 FFAR1 (0.55) FFAR4FFAR1PTPRB
SCHEMBL3578367 0.82 IAPP (0.49) IAPPFFAR4FFAR1ALOX5OR51E2
SCHEMBL31424248 0.82 FFAR1 (0.39) FFAR4FFAR1PTPRB
SCHEMBL30917811 0.81 CYP1A2 (0.53) FFAR4FFAR1CYP1A2CYP2C19
SCHEMBL16840963 0.81 CYP1A2 (0.53) FFAR4FFAR1CYP1A2CYP2C19
SCHEMBL14059359 0.80 MAPT (0.50) FFAR4FFAR1CYP1A2CYP2C19
SCHEMBL12984627 0.79 CYP4F2 (0.56) FFAR4FFAR1
SCHEMBL29021263 0.79 PARP1 (0.36) FFAR4FFAR1KIF11PTPRBCYP1A2
SCHEMBL2302020 0.79 KDM4E (0.47) ALOX5KIF11PTPRBCYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104024250-B Heterocyclic derivatives as Trace Amine Associated Receptors (TAARs) HOFFMAN-LA ROCHE LTD. (CH) 2016-01-27 CN disclosed
CN-104024250-A HETEROCYCLIC DERIVATIVES AS TRACE AMINE ASSOCIATED RECEPTORS (TAARS) HOFFMANN LA ROCHE 2014-09-03 CN disclosed