SCHEMBL28006255

SCHEMBL28006255

O=C(O)Cc1ccnc2ncccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.54
KDM4E B2RXH2 2/20 0.54
MAPT P10636 1/20 0.54
TDP1 Q9NUW8 1/20 0.49
LMNA P02545 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
AKR1B1 P15121 1/20 0.41
NAPRT Q6XQN6 2/20 0.41
EGLN1 Q9GZT9 1/20 0.40
PTGDR2 Q9Y5Y4 8/20 0.40
PRMT5 O14744 1/20 0.40
GABRP O00591 1/20 0.39
GABRD O14764 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA3 P34903 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7992922 0.80 MEN1 (0.48) CYP1A2KDM4EMEN1KMT2A
SCHEMBL5456634 0.80 CYP1A2 (0.67) CYP1A2KDM4EMAPTTDP1LMNA
SCHEMBL15415316 0.79 KDM4E (0.53) KDM4EMAPTTDP1LMNAMEN1
Hydrochloric Acid SCHEMBL3805296 0.79 CYP1A2 (0.65) CYP1A2KDM4EMAPTTDP1LMNA
SCHEMBL3720399 0.79 KDM4E (0.59) CYP1A2KDM4EMAPTTDP1LMNA
Hydrochloric Acid SCHEMBL3712126 0.77 KDM4E (0.57) CYP1A2KDM4EMAPTTDP1LMNA
SCHEMBL8372588 0.77 GSK3A (0.40) KDM4EMAPTTDP1LMNAMEN1
SCHEMBL16361004 0.76 CCR1 (0.51) CYP1A2KDM4EMAPTTDP1LMNA
SCHEMBL9862809 0.76 MAPT (0.46) CYP1A2KDM4EMAPTTDP1LMNA
SCHEMBL10157046 0.75 KDM4E (0.68) CYP1A2KDM4EMAPTTDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104507913-A Antiproliferative benzo[b]azepin-2-ones HOFFMANN LA ROCHE 2015-04-08 CN disclosed