SCHEMBL2800730

SCHEMBL2800730

Clc1cc(C2(Cc3ccccc3)CCN(Cc3ccccc3)C2)cc2cc[nH]c12.Clc1cc(C2(Cc3ccccc3)CCNC2)cc2cc[nH]c12

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 18/20 0.57
SLC6A4 P31645 18/20 0.57
SLC6A3 Q01959 18/20 0.57
CYP2D6 P10635 17/20 0.57
KCNH2 Q12809 5/20 0.57
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.43
KDM4E B2RXH2 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL981123 0.92 KMT2A (0.45) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL985195 0.89 SLC6A2 (0.66) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL984260 0.77 SLC6A2 (0.63) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL984635 0.76 CYP2D6 (0.62) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL982050 0.75 SLC6A2 (0.64) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
5-(3-Benzylpyrrolidin-3-Yl)-1H-Indole (Structural Mix) SCHEMBL982202 0.73 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
5-(3-Benzylpyrrolidin-3-Yl)-1H-Indole (Structural Mix) SCHEMBL982203 0.73 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
5-(3-Benzylpyrrolidin-3-Yl)-1H-Indole (Structural Mix) SCHEMBL982204 0.73 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL983580 0.72 SLC6A2 (0.60) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL980405 0.72 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257545-A1 PYRROLIDINYL DERIVATIVES AND USES THEREOF F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009115427-A1 PYRROLIDINYL DERIVATIVES AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2009-09-24 WO disclosed