SCHEMBL28022117

SCHEMBL28022117

Cc1cc(Nc2cc(N3CCN(C)CC3)nc(S(=O)(=O)Cc3cccc(Cl)c3)n2)[nH]n1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 6/20 0.52
AURKA O14965 9/20 0.48
FLT3 P36888 2/20 0.40
HRH3 Q9Y5N1 1/20 0.39
HTR6 P50406 1/20 0.39
FLT1 P17948 1/20 0.39
KDR P35968 1/20 0.39
AURKB Q96GD4 2/20 0.39
EGFR P00533 1/20 0.39
HTR2C P28335 1/20 0.39
NTRK1 P04629 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28021613 0.93 HRH4 (0.44) HRH4AURKAFLT3HTR6KDR
SCHEMBL28553029 0.91 PIK3CB (0.47) HRH4AURKAAURKB
SCHEMBL28021594 0.91 HRH4 (0.48) HRH4AURKAFLT3HRH3FLT1
SCHEMBL28565380 0.84 HRH4 (0.51) HRH4AURKAAURKBEGFRNTRK1
SCHEMBL2203952 0.81 AURKA (0.57) HRH4AURKAHRH3HTR6AURKB
SCHEMBL28022122 0.81 AURKA (0.46) AURKAFLT3FLT1KDRAURKB
SCHEMBL28562522 0.79 AURKA (0.41) AURKAAURKB
SCHEMBL28562221 0.75 AURKA (0.41) AURKA
SCHEMBL28556719 0.75 AURKA (0.42) AURKA
SCHEMBL2203821 0.73 AURKA (0.64) HRH4AURKAFLT3FLT1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112755193-A Method of treating malignancies with anti-tyrosine kinase inhibitors using dianhydrogalactitol or a derivative thereof 德玛医药 2021-05-07 CN disclosed
CN-104797267-A Method of treating tyrosine kinase inhibitor-resistant malignancies in patients with genetic polymorphism or AHI1 dysregulation or mutation using dianhydrogalactitol, diacetyldianhydrogalactitol, dibromodulcitol, or analogs or derivatives thereof DEL MAR PHARMACEUTICALS 2015-07-22 CN disclosed