SCHEMBL28022736

SCHEMBL28022736

O=C(O)C1CC(F)(F)CCN1C(=O)O

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ACE P12821 4/20 0.31
GRM2 Q14416 1/20 0.31
GRM3 Q14832 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20399718 1.00 ACE (0.31) ACEGRM2GRM3
SCHEMBL15114474 0.81 TSHR (0.38)
SCHEMBL3512916 0.80 GRM2 (0.36) GRM2GRM3
SCHEMBL6919995 0.80 GRM2 (0.36) GRM2GRM3
SCHEMBL4254372 0.80 GRM2 (0.36) GRM2GRM3
SCHEMBL2026722 0.78
SCHEMBL2023665 0.78 CHRM2 (0.31)
SCHEMBL22518862 0.78 CYP2C19 (0.33) GRM2GRM3
SCHEMBL22518863 0.78 CYP2C19 (0.33) GRM2GRM3
SCHEMBL10215476 0.77 HSD17B10 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104940202-B Inhibitors of influenza viruses replication 沃泰克斯药物股份有限公司 2018-10-16 CN disclosed
CN-104940202-A Inhibitors of influenza viruses replication VERTEX PHARMA 2015-09-30 CN disclosed
CN-104922128-A INHIBITORS OF INFLUENZA VIRUSES REPLICATION VERTEX PHARMA 2015-09-23 CN disclosed
CN-102458408-B Inhibitors of influenza virus replication VERTEX PHARMA 2015-06-03 CN disclosed