SCHEMBL28027989

SCHEMBL28027989

CC1C(=O)C(c2ccccc2)CN1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
KMT2A Q03164 1/20 0.47
BRD4 O60885 3/20 0.43
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 2/20 0.41
SLC6A3 Q01959 2/20 0.41
SRD5A1 P18405 1/20 0.41
ATM Q13315 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HTR1A P08908 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
MAPK1 P28482 1/20 0.38
THPO P40225 1/20 0.38
HIF1A Q16665 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11618119 0.79 SLC6A2 (0.53) TSHRKMT2ABRD4SLC6A2SLC6A4
SCHEMBL28027961 0.75 TSHR (0.44) TSHRKMT2A
SCHEMBL27262808 0.71 TSHR (0.56) TSHRKMT2ABRD4SLC6A2SLC6A4
SCHEMBL28028150 0.71 SLC6A2 (0.46) KMT2ASLC6A2SLC6A4SLC6A3ATM
SCHEMBL5246352 0.70 SLC6A2 (0.57) SLC6A2SLC6A4SLC6A3ALDH1A1MAPK1
SCHEMBL5309449 0.69 SLC6A2 (0.45) SLC6A2SLC6A4SLC6A3MAPK1
SCHEMBL11645243 0.69 DRD1 (0.56) SLC6A2SLC6A4SLC6A3SMN1; SMN2MAPK1
SCHEMBL10883366 0.69 BRD4 (0.50) TSHRKMT2ABRD4SLC6A2SLC6A4
SCHEMBL10258633 0.69 SLC6A2 (0.44) TSHRKMT2ABRD4SLC6A2SLC6A4
SCHEMBL11619884 0.68 SLC6A2 (0.55) TSHRKMT2ASLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104854108-A Pyrrolotriazinone derivatives as pi3k inhibitors ALMIRALL SA 2015-08-19 CN claimed
CN-104854108-A Pyrrolotriazinone derivatives as pi3k inhibitors ALMIRALL SA 2015-08-19 CN disclosed