SCHEMBL28028400

SCHEMBL28028400

COC(=O)c1cccc(OCC(F)F)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 2/20 0.56
KDM4E B2RXH2 1/20 0.55
CYSLTR1 Q9Y271 1/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
USP2 O75604 1/20 0.51
LMNA P02545 1/20 0.51
MAPK1 P28482 1/20 0.51
HSD17B10 Q99714 1/20 0.51
NPC1 O15118 1/20 0.50
POLB P06746 1/20 0.50
RAB9A P51151 1/20 0.50
BLM P54132 1/20 0.50
TP53 P04637 1/20 0.49
LOXL2 Q9Y4K0 1/20 0.49
CYP4F2 P78329 1/20 0.48
CYP4A11 Q02928 1/20 0.48
VDR P11473 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
NR1H4 Q96RI1 1/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26049008 0.86 NR1H4 (0.60) MRGPRX4KDM4ECYSLTR1SMN1; SMN2USP2
SCHEMBL7988758 0.85 KDM4E (0.62) MRGPRX4KDM4ECYSLTR1SMN1; SMN2USP2
SCHEMBL3239119 0.85 MRGPRX4 (0.53) MRGPRX4KDM4ECYSLTR1SMN1; SMN2NPC1
SCHEMBL17416724 0.85 TDP1 (0.41) MRGPRX4KDM4EL3MBTL1NR1H4
SCHEMBL24763747 0.84 KDM4E (0.54) MRGPRX4KDM4ECYSLTR1SMN1; SMN2USP2
SCHEMBL6780356 0.84 KDM4E (0.54) MRGPRX4KDM4ECYSLTR1SMN1; SMN2USP2
SCHEMBL2947246 0.83 NR4A2 (0.59) MRGPRX4CYSLTR1NPC1RAB9ANR1H4
SCHEMBL30281398 0.83 NR4A2 (0.59) MRGPRX4CYSLTR1NPC1RAB9ANR1H4
SCHEMBL27439509 0.83 MRGPRX4 (0.59) MRGPRX4KDM4ECYSLTR1SMN1; SMN2MAPK1
SCHEMBL14896697 0.82 KDM4E (0.53) MRGPRX4KDM4ECYSLTR1SMN1; SMN2USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104812755-A Pyrazolopyridine derivatives as TTX-S blockers RAQUALIA PHARMA INC 2015-07-29 CN disclosed