SCHEMBL28028753

SCHEMBL28028753

CNc1ccccc1.Fc1cccnc1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.52
NAPRT Q6XQN6 1/20 0.39
KCNH2 Q12809 2/20 0.39
AURKA O14965 2/20 0.36
KDM1A O60341 2/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
ATM Q13315 1/20 0.35
MAOA P21397 2/20 0.34
MAOB P27338 2/20 0.34
DHODH Q02127 1/20 0.34
PLK4 O00444 1/20 0.34
PDPK1 O15530 1/20 0.34
JAK2 O60674 1/20 0.34
PRKD3 O94806 1/20 0.34
MAP4K4 O95819 1/20 0.34
NTRK1 P04629 1/20 0.34
INSR P06213 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL255507 0.79
SCHEMBL29457380 0.79
Hydrochloric Acid SCHEMBL29195521 0.77
Hydrochloric Acid SCHEMBL34460386 0.77
SCHEMBL30534895 0.77
SCHEMBL4057572 0.77
Lithium SCHEMBL4057575 0.77
Pyridine SCHEMBL29035748 0.72 NAPRT (0.44) TSHRNAPRTKDM4ENPC1RAB9A
Hydrochloric Acid SCHEMBL5440963 0.72 TSHR (0.88) TSHRNAPRTKDM1AKDM4EKMT2A
Hydrochloric Acid SCHEMBL27706419 0.72 TSHR (0.88) TSHRNAPRTKDM1AKDM4ECLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104995198-A POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES INC 2015-10-21 CN disclosed