SCHEMBL28032955

SCHEMBL28032955

NC(C(=O)O)[C@@H](Cc1cc(F)c(F)cc1F)C(=O)OCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 12/20 0.51
SLC1A1 P43005 5/20 0.48
SLC1A3 P43003 3/20 0.48
SLC1A2 P43004 3/20 0.48
MEN1 O00255 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 1/20 0.41
CYP3A4 P08684 1/20 0.41
SLC15A1 P46059 1/20 0.40
LTA4H P09960 1/20 0.40
LAP3 P28838 1/20 0.40
DPP7 Q9UHL4 4/20 0.40
DPP8 Q6V1X1 3/20 0.40
DPP9 Q86TI2 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11232982 1.00 DPP4 (0.51) DPP4SLC1A1SLC1A3SLC1A2MEN1
SCHEMBL27943329 1.00 DPP4 (0.51) DPP4SLC1A1SLC1A3SLC1A2MEN1
SCHEMBL19500639 0.79 DPP4 (0.62) DPP4CYP3A4SLC15A1DPP7DPP8
SCHEMBL19500635 0.79 DPP4 (0.62) DPP4CYP3A4SLC15A1DPP7DPP8
SCHEMBL11190716 0.78 SLC1A1 (0.54) SLC1A1SLC1A3SLC1A2MEN1CYP1A2
SCHEMBL29619670 0.78 DPP4 (0.49) DPP4ALDH1A1CYP3A4LTA4HLAP3
SCHEMBL28055243 0.77 DPP4 (0.49) DPP4SLC1A1SLC1A3SLC1A2CYP3A4
SCHEMBL11221173 0.77 DPP4 (0.49) DPP4SLC1A1SLC1A3SLC1A2CYP3A4
SCHEMBL27899116 0.77 DPP4 (0.49) DPP4SLC1A1SLC1A3SLC1A2CYP3A4
SCHEMBL27501469 0.77 SLC1A1 (0.56) SLC1A1SLC1A3SLC1A2MEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105294479-A Preparation method of 3R-amino substituted butyrylamide derivative XINFA PHARMACEUTICAL CO LTD 2016-02-03 CN disclosed
CN-105061434-A Low-cost preparation method of sitagliptin phosphate XINFA PHARMACEUTICAL CO LTD 2015-11-18 CN disclosed