SCHEMBL28034335

SCHEMBL28034335

CCOc1ccc(C(=O)O)cc1OCC1CC1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.64
POLB P06746 1/20 0.59
CASP6 P55212 1/20 0.59
LMNA P02545 1/20 0.53
PDE4B Q07343 8/20 0.51
PDE4A P27815 3/20 0.51
PDE4C Q08493 3/20 0.51
PDE4D Q08499 3/20 0.51
GLA P06280 1/20 0.49
NPSR1 Q6W5P4 1/20 0.48
APOBEC3G Q9HC16 1/20 0.48
MAPK1 P28482 1/20 0.48
RXRA P19793 1/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
ALOX15 P16050 1/20 0.47
MRGPRX4 Q96LA9 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28034346 0.93 PDE4B (0.53) TSHRPOLBCASP6PDE4BPDE4A
SCHEMBL28034364 0.87 MAPK1 (0.65) TSHRPDE4BPDE4APDE4CPDE4D
SCHEMBL29670247 0.87 TSHR (0.66) TSHRLMNAPDE4BPDE4APDE4C
SCHEMBL15596058 0.87 TSHR (0.66) TSHRLMNAPDE4BPDE4APDE4C
SCHEMBL30575456 0.87 CA12 (0.63) TSHRPDE4BPDE4APDE4CPDE4D
SCHEMBL1031663 0.87 CA12 (0.63) TSHRPDE4BPDE4APDE4CPDE4D
SCHEMBL29882038 0.86 TSHR (0.83) TSHRPOLBCASP6LMNANPSR1
SCHEMBL177424 0.86 TSHR (0.83) TSHRPOLBCASP6LMNANPSR1
SCHEMBL28033773 0.86 PDE4B (0.55) TSHRPDE4BPDE4APDE4CPDE4D
SCHEMBL14799306 0.83 TSHR (0.47) TSHRPOLBCASP6PDE4BPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105085429-B Aromatic heterocyclic derivative and application thereof in medicines 广东东阳光药业有限公司 2019-12-10 CN disclosed
CN-105085429-A Heteroaromatic derivative and application thereof to medicament GUANGDONG HEC PHARMACEUTICAL 2015-11-25 CN disclosed