SCHEMBL28037156

SCHEMBL28037156

C#Cc1ccc(C2CCCN2)c(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HTR2C P28335 3/20 0.36
HTR2A P28223 2/20 0.36
HTR2B P41595 2/20 0.36
AR P10275 4/20 0.33
ADORA2A P29274 5/20 0.32
ADORA1 P30542 5/20 0.32
CYP3A4 P08684 3/20 0.32
KCNH2 Q12809 3/20 0.32
ADORA3 P0DMS8 2/20 0.32
ADORA2B P29275 1/20 0.32
CYP2C19 P33261 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NR1I2 O75469 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.32
HTR1A P08908 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11224505 0.78 HTR2C (0.41) HTR2CHTR2AHTR2BARCYP3A4
SCHEMBL29484307 0.77 HTR2C (0.56) MEN1KMT2AHTR2CHTR2BHTR1A
SCHEMBL457401 0.77 HTR2C (0.56) MEN1KMT2AHTR2CHTR2BHTR1A
SCHEMBL29589456 0.77 HTR2C (0.56) MEN1KMT2AHTR2CHTR2BHTR1A
SCHEMBL11234509 0.77 HTR2C (0.41) HTR2CARCYP3A4KCNH2CYP2C19
SCHEMBL11239231 0.77 HTR2C (0.41) HTR2CARCYP3A4KCNH2CYP2C19
Hydrochloric Acid SCHEMBL31444282 0.76 HTR2C (0.57) MEN1KMT2AHTR2CHTR2AHTR2B
Hydrochloric Acid SCHEMBL6092900 0.76 HTR2C (0.57) MEN1KMT2AHTR2CHTR2AHTR2B
SCHEMBL932518 0.74 MEN1 (0.39) MEN1KMT2AHTR2CHTR2AKCNH2
SCHEMBL454693 0.74 MEN1 (0.39) MEN1KMT2AHTR2CHTR2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105061326-A Pyridazinone derivatives as well as preparation method and application thereof SICHUAN BAILI PHARMACEUTICAL CO LTD 2015-11-18 CN disclosed