SCHEMBL28037333

SCHEMBL28037333

CC(C)(C)OC(=O)N1Cc2cn(CS(C)(=O)=O)nc2C1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.40
HDAC1 Q13547 1/20 0.39
ESR2 Q92731 1/20 0.38
MAPK1 P28482 1/20 0.38
NAMPT P43490 1/20 0.37
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
MAPT P10636 1/20 0.36
GPR119 Q8TDV5 7/20 0.36
SLC34A1 Q06495 1/20 0.36
SLC6A9 P48067 1/20 0.36
KCNH2 Q12809 1/20 0.36
STS P08842 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31460333 0.86 HDAC1 (0.41) NR1H2HDAC1ESR2MAPK1NAMPT
SCHEMBL20738563 0.86 HDAC1 (0.41) NR1H2HDAC1ESR2MAPK1NAMPT
SCHEMBL9918101 0.84 HDAC1 (0.40) NR1H2HDAC1ESR2MAPK1NAMPT
SCHEMBL28036918 0.84 HDAC1 (0.40) NR1H2HDAC1ESR2MAPK1NAMPT
SCHEMBL20392575 0.82 HDAC1 (0.43) NR1H2HDAC1ESR2MAPK1NAMPT
SCHEMBL12451984 0.82 HDAC1 (0.39) NR1H2HDAC1ESR2MAPK1NAMPT
SCHEMBL6893628 0.82 NR1H2 (0.40) NR1H2HDAC1ESR2MAPK1NAMPT
SCHEMBL14358443 0.82 HDAC1 (0.40) NR1H2HDAC1ESR2MAPK1NAMPT
SCHEMBL23372983 0.81 HDAC1 (0.46) NR1H2HDAC1ESR2MAPK1NAMPT
SCHEMBL24506914 0.81 SLC34A1 (0.46) NR1H2HDAC1ESR2MAPK1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105037367-A Amino six-membered ring derivative and application thereof in medicines SICHUAN HAISCO PHARMACEUTICAL CO LTD 2015-11-11 CN disclosed