SCHEMBL28037875

SCHEMBL28037875

CCN1CCN(c2nc(NCc3ccc(-c4ccccc4N)cc3)c3ncn(C4CCCC4)c3n2)CC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 12/20 0.63
CCNE1 P24864 10/20 0.63
CDK2 P24941 10/20 0.63
CDK5 Q00535 2/20 0.55
CCNE2 O96020 3/20 0.51
CCNA2 P20248 2/20 0.51
CCNA1 P78396 2/20 0.51
CSNK1E P49674 2/20 0.50
CLK1 P49759 2/20 0.50
CLK2 P49760 2/20 0.50
CDK7 P50613 2/20 0.50
DYRK1A Q13627 2/20 0.50
CLK4 Q9HAZ1 2/20 0.50
CTSL P07711 1/20 0.49
TDP1 Q9NUW8 1/20 0.48
PDGFRA P16234 1/20 0.48
CCNB2 O95067 1/20 0.47
CDK4 P11802 1/20 0.47
CCNB1 P14635 1/20 0.47
CCND1 P24385 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17352589 0.92 CDK1 (0.65) CDK1CCNE1CDK2CDK5CCNE2
SCHEMBL15941141 0.91 CDK1 (0.62) CDK1CCNE1CDK2CDK5CCNE2
SCHEMBL28037848 0.91 CDK1 (0.62) CDK1CCNE1CDK2CDK5CCNE2
SCHEMBL28038208 0.90 CDK1 (0.64) CDK1CCNE1CDK2CDK5CCNE2
SCHEMBL15941368 0.89 CDK1 (0.65) CDK1CCNE1CDK2CDK5CCNE2
SCHEMBL17352540 0.89 CDK1 (0.65) CDK1CCNE1CDK2CDK5CCNE2
SCHEMBL15941014 0.87 CDK1 (0.58) CDK1CCNE1CDK2CDK5CCNE2
SCHEMBL28037886 0.83 CDK1 (0.62) CDK1CCNE1CDK2CDK5CCNE2
SCHEMBL28037850 0.83 CDK1 (0.63) CDK1CCNE1CDK2CDK5CSNK1E
SCHEMBL15940975 0.82 CDK1 (0.62) CDK1CCNE1CDK2CDK5CCNE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105026396-A 2-substituted-6-biarylmethylamino-9-cyclopentyl-9h-purine derivatives, use thereof as medicaments, and pharmaceutical compositions UNIV PALACKEHO 2015-11-04 CN disclosed