SCHEMBL28038987

SCHEMBL28038987

Nc1cc(Nc2ccncn2)ncn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.54
CDK5 Q00535 2/20 0.50
GSK3A P49840 1/20 0.50
CDK9 P50750 1/20 0.50
TAOK1 Q7L7X3 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50
CDK1 P06493 1/20 0.46
CCNB1 P14635 1/20 0.46
CCNA2 P20248 1/20 0.46
CCNE1 P24864 1/20 0.46
CDK2 P24941 1/20 0.46
CDK5R1 Q15078 1/20 0.46
SCN9A Q15858 1/20 0.44
KDR P35968 3/20 0.43
PIK3C3 Q8NEB9 2/20 0.42
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
TYK2 P29597 1/20 0.42
MKNK1 Q9BUB5 6/20 0.41
HRH4 Q9H3N8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4630887 0.83 GSK3A (0.53) HSP90AA1CDK5GSK3ACDK9TAOK1
Hydrochloric Acid SCHEMBL7857018 0.81 GSK3A (0.51) HSP90AA1CDK5GSK3ACDK9TAOK1
SCHEMBL28038743 0.81 CDK5 (0.58) HSP90AA1CDK5TAOK1CLK4CDK1
SCHEMBL16916919 0.74 JAK2 (0.52) CDK5GSK3ACDK9TAOK1CLK4
SCHEMBL16996884 0.74 GSK3A (0.48) CDK5GSK3ACDK9TAOK1CLK4
SCHEMBL29919700 0.74 SCN9A (0.53) CDK5CDK1CCNB1CCNA2CCNE1
SCHEMBL31247573 0.74 KDM4E (0.57) CDK5GSK3ACDK9CLK4CDK1
SCHEMBL28936140 0.74 SCN9A (0.53) CDK5CDK1CCNB1CCNA2CCNE1
SCHEMBL27606961 0.74 GSK3A (0.48) CDK5GSK3ACDK9TAOK1CLK4
SCHEMBL4666187 0.73 RAD52 (0.59) HSP90AA1KDRMKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105051030-A Diaminoheteroaryl substituted indazoles Bayer Pharma AG 2015-11-11 CN claimed
CN-105051030-A Diaminoheteroaryl substituted indazoles Bayer Pharma AG 2015-11-11 CN disclosed