SCHEMBL28039002

SCHEMBL28039002

FCCn1ccnc1-c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.64
PLAA Q9Y263 1/20 0.46
ALPG P10696 1/20 0.45
PDE6D O43924 4/20 0.43
CYP3A4 P08684 2/20 0.42
CYP2C19 P33261 2/20 0.42
TSHR P16473 1/20 0.42
CYP2C9 P11712 1/20 0.42
HIF1A Q16665 1/20 0.42
BRD4 O60885 1/20 0.42
LIMK2 P53671 1/20 0.41
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA3 P07451 1/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1306747 0.86 ESR1 (0.69) ESR1PLAAALPGPDE6DCYP3A4
SCHEMBL7095574 0.85 ESR1 (0.68) ESR1PLAAALPGPDE6DCYP3A4
Hydrochloric Acid SCHEMBL10366282 0.84 ESR1 (0.67) ESR1PLAAALPGPDE6DCYP3A4
SCHEMBL462620 0.83 ESR1 (0.60) ESR1PLAAALPGPDE6DCYP3A4
SCHEMBL17219702 0.82 ESR1 (0.64) ESR1PLAAALPGPDE6DCYP3A4
SCHEMBL20083767 0.82 ESR1 (0.64) ESR1PLAAALPGPDE6DCYP3A4
SCHEMBL9444420 0.82 ESR1 (0.64) ESR1PLAAALPGPDE6DCYP3A4
SCHEMBL5662079 0.82 ESR1 (0.69) ESR1PLAAALPGPDE6DCYP3A4
SCHEMBL27850097 0.81 ESR1 (0.58) ESR1PLAAALPGPDE6DCYP3A4
SCHEMBL8910757 0.81 ESR1 (0.59) ESR1PLAAALPGPDE6DCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105164125-B 2-phenyl or 2-heteroaryl imidazo [1,2-a ] pyridine derivatives 豪夫迈·罗氏有限公司 2017-10-13 CN claimed
CN-105164125-A 2-phenyl or 2-heteroaryl imidazo [1, 2-a ] pyridine derivatives HOFFMANN LA ROCHE 2015-12-16 CN claimed
CN-105164125-B 2-phenyl or 2-heteroaryl imidazo [1,2-a ] pyridine derivatives 豪夫迈·罗氏有限公司 2017-10-13 CN disclosed
CN-105164125-A 2-phenyl or 2-heteroaryl imidazo [1, 2-a ] pyridine derivatives HOFFMANN LA ROCHE 2015-12-16 CN disclosed