SCHEMBL28039439

SCHEMBL28039439

CSc1ncc(CO)c(Nc2cccc(N)c2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.52
SYK P43405 4/20 0.47
MAPK1 P28482 1/20 0.47
AHR P35869 1/20 0.40
SRC P12931 3/20 0.39
EGFR P00533 2/20 0.39
ABL1 P00519 2/20 0.39
BCR P11274 2/20 0.39
TOP2A P11388 1/20 0.39
PRKACA P17612 1/20 0.39
PRKACG P22612 1/20 0.39
PRKACB P22694 1/20 0.39
BRD4 O60885 1/20 0.39
MAPT P10636 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
GFER P55789 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4712352 0.85 HTT (0.51) HTTSYKMAPK1SRCABL1
SCHEMBL6617756 0.84 HTT (0.54) HTTSYKMAPK1SRCEGFR
SCHEMBL24668609 0.84 CDK1 (0.47) HTTSYKMAPK1SRCEGFR
SCHEMBL15992691 0.83 HTT (0.51) HTTSYKMAPK1EGFRBRD4
SCHEMBL30069455 0.82 HTT (0.53) HTTSYKMAPK1EGFRMAPT
SCHEMBL28382393 0.82 HTT (0.53) HTTSYKMAPK1EGFRMAPT
SCHEMBL30596936 0.81 HTT (0.47) HTTSYKMAPK1KMT2AKDM4E
SCHEMBL26107898 0.81 HTT (0.47) HTTSYKMAPK1KMT2AKDM4E
SCHEMBL16003515 0.79 SYK (0.47) HTTSYKMAPK1AHRSRC
SCHEMBL29497529 0.78 SYK (0.54) HTTSYKMAPK1EGFRBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104968664-A BICYCLIC COMPOUND FUNCTIONING AS TYROSINE KINASE INHIBITOR KBP BIOSCIENCES CO LTD 2015-10-07 CN disclosed