SCHEMBL28040096

SCHEMBL28040096

NC(=O)c1cc(C(=O)N2CCOCC2)cc2[nH]c3ccccc3c12

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 17/20 0.54
JAK1 P23458 7/20 0.54
TYK2 P29597 7/20 0.54
JAK3 P52333 7/20 0.54
BTK Q06187 6/20 0.48
POLB P06746 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27997777 0.84 JAK2 (0.71) JAK2JAK1TYK2JAK3BTK
SCHEMBL27998021 0.81 JAK2 (0.61) JAK2JAK1TYK2JAK3BTK
SCHEMBL27998017 0.81 JAK2 (0.50) JAK2JAK1TYK2JAK3BTK
SCHEMBL15995152 0.79 JAK2 (0.56) JAK2JAK1TYK2JAK3BTK
SCHEMBL28258694 0.79 MAPK10 (0.45) JAK2JAK1TYK2JAK3POLB
SCHEMBL28816460 0.79 JAK2 (0.53) JAK2JAK1TYK2JAK3BTK
SCHEMBL148196 0.75 JAK2 (0.58) JAK2JAK1TYK2JAK3BTK
SCHEMBL27997807 0.75 JAK2 (0.59) JAK2JAK1TYK2JAK3BTK
SCHEMBL148776 0.74 JAK2 (0.53) JAK2JAK1TYK2JAK3
SCHEMBL27997819 0.73 JAK2 (0.60) JAK2JAK1TYK2JAK3BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105008352-B Carbazole compounds useful as bromodomain inhibitors 百时美施贵宝公司 2018-12-07 CN disclosed
CN-105008352-A Carbazole compounds useful as bromodomain inhibitors BRISTOL MYERS SQUIBB CO 2015-10-28 CN disclosed