SCHEMBL28045774

SCHEMBL28045774

COc1ncc(CCBr)cc1-c1cccc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 4/20 0.44
CTSA P10619 2/20 0.44
NR1I3 Q14994 1/20 0.40
PDE4D Q08499 2/20 0.39
PDE4A P27815 1/20 0.39
PDE4C Q08493 1/20 0.39
FYN P06241 2/20 0.39
FFAR4 Q5NUL3 1/20 0.38
DHFR P00374 1/20 0.38
NUDT1 P36639 1/20 0.38
NOTUM Q6P988 1/20 0.37
KMT2A Q03164 1/20 0.37
CCR4 P51679 1/20 0.37
HRH1 P35367 1/20 0.36
KDR P35968 1/20 0.36
EPHB4 P54760 1/20 0.36
TEK Q02763 1/20 0.36
MET P08581 1/20 0.36
AXL P30530 1/20 0.36
MERTK Q12866 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16045821 0.90 PDE4B (0.46) PDE4BCTSANR1I3PDE4DPDE4A
SCHEMBL16112949 0.85 PDE4B (0.46) PDE4BCTSANR1I3PDE4DPDE4A
SCHEMBL16114574 0.84 PDE4B (0.46) PDE4BCTSANR1I3PDE4DPDE4A
SCHEMBL16114185 0.84 CTSA (0.48) PDE4BCTSANR1I3PDE4DPDE4A
SCHEMBL28045842 0.84 PDE4B (0.42) PDE4BCTSADHFRNUDT1HRH1
SCHEMBL16045964 0.82 PDE4B (0.44) PDE4BCTSANR1I3PDE4DPDE4A
SCHEMBL16114578 0.82 PDE4B (0.44) PDE4BCTSANR1I3PDE4DPDE4A
SCHEMBL16075859 0.82 CTSA (0.48) PDE4BCTSANR1I3PDE4DPDE4A
SCHEMBL16044652 0.81 PDE4B (0.43) PDE4BCTSANR1I3PDE4DPDE4A
SCHEMBL16043956 0.81 CTSA (0.45) PDE4BCTSANR1I3PDE4DPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143207-A Substituted pyridine and substituted pyrazine compounds as PDE4 inhibitors DART NEUROSCIENCE LLC 2015-12-09 CN disclosed