SCHEMBL28048281

SCHEMBL28048281

CC(OC(=O)Cl)c1cccc(F)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
MTOR P42345 1/20 0.41
KDM4E B2RXH2 1/20 0.41
AOC3 Q16853 1/20 0.41
HPGD P15428 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
SLC6A4 P31645 1/20 0.40
LMNA P02545 1/20 0.39
CNR2 P34972 1/20 0.39
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
OPRM1 P35372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19881211 0.85 HDAC4 (0.47) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL27427626 0.85 HDAC4 (0.47) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL27795851 0.83 HDAC4 (0.46) HDAC4HDAC7HDAC5CES2CES1
Hydrochloric Acid SCHEMBL27533449 0.80 HDAC4 (0.43) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL28165650 0.78 AOC3 (0.43) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL8823897 0.78 HCAR2 (0.58) KMT2ALMNAOPRM1
SCHEMBL5692198 0.78 HCAR2 (0.58) KMT2ALMNAOPRM1
SCHEMBL8823875 0.78 HCAR2 (0.58) KMT2ALMNAOPRM1
SCHEMBL8498061 0.77 HDAC4 (0.50) HDAC4HDAC7HDAC5CES2CES1
SCHEMBL3883489 0.77 HDAC4 (0.42) HDAC4HDAC7HDAC5CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105142640-B Tyrosine protein kinase inhibitor 豪夫迈·罗氏有限公司 2017-08-29 CN disclosed
CN-105142640-A Inhibitors of bruton's tyrosine kinase HOFFMANN LA ROCHE 2015-12-09 CN disclosed