SCHEMBL28048683

SCHEMBL28048683

CN1CCN(C(=O)N2CCN(C)[C@@H](CO)C2)C[C@@H]1CO

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.40
CA2 P00918 4/20 0.40
CA4 P22748 4/20 0.40
CA9 Q16790 4/20 0.40
POLB P06746 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 2/20 0.33
PRKCB P05771 1/20 0.32
CYP1A2 P05177 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
CHRM1 P11229 1/20 0.31
TACR1 P25103 1/20 0.31
GAA P10253 2/20 0.31
MGAM O43451 1/20 0.31
SMYD3 Q9H7B4 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3830521 0.86 CA1 (0.39) CA1CA2CA4CA9POLB
SCHEMBL25308860 0.86 CA1 (0.39) CA1CA2CA4CA9POLB
SCHEMBL12439869 0.86 CYP1A2 (0.43) CA1CA2CA4CA9POLB
SCHEMBL14433125 0.86 CYP1A2 (0.43) CA1CA2CA4CA9POLB
SCHEMBL2015636 0.86 CA1 (0.39) CA1CA2CA4CA9POLB
SCHEMBL8321488 0.82 HTT (0.45) CA1CA2CA4CA9ALDH1A1
SCHEMBL16838110 0.82 HTT (0.45) CA1CA2CA4CA9ALDH1A1
SCHEMBL25587621 0.82 CA1 (0.36) CA1CA2CA4CA9POLB
SCHEMBL305616 0.78 NR1H2 (0.51) ALDH1A1RECQL
SCHEMBL2157286 0.78 NR1H2 (0.51) ALDH1A1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105377851-A BET bromodomain inhibitors and therapeutic methods using these inhibitors UNIV MICHIGAN REGENTS 2016-03-02 CN disclosed