SCHEMBL28048782

SCHEMBL28048782

O=COc1ccc2c(ccn2C(=O)O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 1/20 0.43
TFPI2 P48307 3/20 0.41
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
OXER1 Q8TDS5 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.35
TSHR P16473 1/20 0.35
RAB9A P51151 1/20 0.35
ACHE P22303 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3249823 0.81 TUBB1 (0.62) TUBB1TFPI2HDAC1HDAC6L3MBTL1
SCHEMBL2651525 0.77 PIM1 (0.47) TUBB1TFPI2KDM4EPPARDPPARA
SCHEMBL28264551 0.76 CYP2A6 (0.34) TUBB1L3MBTL1POLBHTR6PLA2G4A
SCHEMBL15969044 0.76 CYP2A6 (0.57) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5483649 0.74 SRD5A2 (0.57) HDAC1HDAC6RAB9AKDM4EALDH1A1
SCHEMBL2795863 0.73 KDR (0.45) TUBB1
SCHEMBL28048800 0.73 CHEK1 (0.42) RAB9AKDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL30063197 0.73 ELANE (0.47) TUBB1TFPI2OXER1L3MBTL1TSHR
SCHEMBL25857593 0.72 HTR2C (0.39) TUBB1TFPI2L3MBTL1POLBHTR6
SCHEMBL26432938 0.72 CYP2A6 (0.35) TUBB1TFPI2L3MBTL1POLBHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105188696-A Gamma-diketones as WNT/beta -catenin signaling pathway activators SAMUMED LLC 2015-12-23 CN disclosed