2-Chloropyridine

2-Chloropyridine

SCHEMBL28051574

Clc1ccccn1.O=C(O)O.[CsH]

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of 2-Chloropyridine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.73
LMNA P02545 2/20 0.50
NAPRT Q6XQN6 2/20 0.50
P4HTM Q9NXG6 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
KMT2A Q03164 2/20 0.45
GRM5 P41594 1/20 0.44
SMARCA2 P51531 1/20 0.44
SMARCA4 P51532 1/20 0.44
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
PKM P14618 1/20 0.42
TLR7 Q9NYK1 1/20 0.41
PTGS2 P35354 1/20 0.41
KCNQ3 O43525 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
2-Chloropyridine SCHEMBL7769567 0.98 TDP1 (0.76) TDP1LMNANAPRTP4HTML3MBTL1
2-Chloropyridine SCHEMBL5718309 0.91 TDP1 (0.73) TDP1LMNANAPRTP4HTML3MBTL1
2-Chloropyridine SCHEMBL28789823 0.88 TDP1 (0.76) TDP1LMNANAPRTP4HTML3MBTL1
2-Chloropyridine SCHEMBL27450572 0.85
2-Chloropyridine SCHEMBL28283275 0.85 TDP1 (1.00) TDP1LMNAP4HTML3MBTL1CES2
2-Chloropyridine SCHEMBL10690176 0.85 TDP1 (1.00) TDP1LMNAP4HTML3MBTL1CES2
2-Chloropyridine SCHEMBL16637 0.85
2-Chloropyridine SCHEMBL11389784 0.85
2-Chloropyridine SCHEMBL29402311 0.85
2-Chloropyridine SCHEMBL28051573 0.84 TDP1 (0.70) TDP1LMNANAPRTP4HTML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105324376-B Heteroaromatics and its purposes as dopamine D 1 part 辉瑞大药厂 2017-06-23 CN disclosed
CN-105324376-A Heteroaromatic compounds and their use as dopamine d1 ligands PFIZER 2016-02-10 CN disclosed