SCHEMBL28051992

SCHEMBL28051992

NC(=O)c1cc(-c2cnccn2)ccn1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.59
TSHR P16473 1/20 0.59
MC4R P32245 1/20 0.59
ADRA1A P35348 1/20 0.59
MC3R P41968 1/20 0.59
PIM2 Q9P1W9 2/20 0.50
PIM1 P11309 1/20 0.49
HDAC3 O15379 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC2 Q92769 2/20 0.46
CYP11B2 P19099 1/20 0.45
GSK3B P49841 1/20 0.45
KDM4E B2RXH2 1/20 0.43
NAPRT Q6XQN6 1/20 0.43
HCAR2 Q8TDS4 1/20 0.43
PIK3CD O00329 1/20 0.42
PIK3CA P42336 1/20 0.42
PIK3CB P42338 1/20 0.42
PI4KA P42356 1/20 0.42
PIK3CG P48736 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30839465 0.78 CHEK2 (0.49) KDM4ENAPRTBAZ2B
Hydrochloric Acid SCHEMBL9792812 0.78 MKNK1 (0.52) ADORA3TSHRMC4RADRA1AMC3R
Pyrazinamide SCHEMBL27455922 0.78
SCHEMBL29516759 0.77 CHUK (0.56) ADORA3TSHRMC4RADRA1AMC3R
SCHEMBL933914 0.77 MKNK1 (0.59) ADORA3TSHRMC4RADRA1AMC3R
SCHEMBL30761107 0.77 MKNK1 (0.59) ADORA3TSHRMC4RADRA1AMC3R
SCHEMBL20169521 0.76 PIK3CD (0.46) PIM2PIM1HDAC3HDAC1HDAC2
SCHEMBL2735065 0.76 MKNK1 (0.57) ADORA3TSHRMC4RADRA1AMC3R
SCHEMBL29355955 0.76 MKNK1 (0.57) ADORA3TSHRMC4RADRA1AMC3R
Pyrazinamide SCHEMBL18364991 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658639-A Alkynyl alcohols and methods of use 豪夫迈·罗氏有限公司 2016-06-08 CN disclosed