SCHEMBL28052081

SCHEMBL28052081

COc1cc2c([nH]c(=O)c3scc(Br)c32)c(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NEK1 Q96PY6 14/20 0.38
PDE3B Q13370 3/20 0.37
PDE3A Q14432 3/20 0.37
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2B Q13224 1/20 0.36
GRIN2C Q14957 1/20 0.36
GRIN3A Q8TCU5 1/20 0.36
MAOA P21397 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2552572 0.76 NEK1 (0.52) NEK1
SCHEMBL16858750 0.68 NEK1 (0.38) NEK1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL1429394 0.66 PRKDC (0.39) PDE3BPDE3AGRIN2DGRIN3BGRIN1
SCHEMBL2549746 0.66 NEK1 (0.63) NEK1
SCHEMBL2553600 0.64 NEK1 (0.47) NEK1
SCHEMBL2547614 0.63 CHEK1 (0.43) NEK1KDM4EALDH1A1HPGD
SCHEMBL16858741 0.63 PARP1 (0.41) NEK1GRIN2DGRIN3BGRIN1GRIN2A
Hydrochloric Acid SCHEMBL15092557 0.62 CHEK1 (0.42) NEK1KDM4EALDH1A1HPGD
SCHEMBL2552389 0.61 NEK1 (0.60) NEK1
SCHEMBL2553281 0.60 CYP1A2 (0.52) KDM4EALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102917590-B Tricyclic compound and the PBK inhibitor containing described compound ONCOTHERAPY SCIENCE, INC. (JP) 2016-02-17 CN disclosed