SCHEMBL28053591

SCHEMBL28053591

O=C(c1cnc(N2CCOCC2)nc1)c1cnc(N2CCOCC2)nc1

nearest known ligand 0.77

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.77
HDAC6 Q9UBN7 1/20 0.51
ALDH1A1 P00352 3/20 0.50
ADRA1A P35348 1/20 0.48
KDM4E B2RXH2 3/20 0.47
HPGD P15428 1/20 0.47
ALOX15 P16050 1/20 0.47
HSD17B10 Q99714 1/20 0.47
HTT P42858 1/20 0.46
PIK3CA P42336 4/20 0.45
PIK3R1 P27986 3/20 0.45
MTOR P42345 3/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CNR2 P34972 1/20 0.44
MAPK1 P28482 1/20 0.44
PTPN11 Q06124 1/20 0.44
KMT2A Q03164 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL605729 0.87 POLB (1.00) POLBHDAC6ALDH1A1ADRA1AKDM4E
SCHEMBL12647466 0.86 POLB (0.73) POLBHDAC6ALDH1A1ADRA1AKDM4E
SCHEMBL3126575 0.86 POLB (0.73) POLBHDAC6ALDH1A1ADRA1AKDM4E
SCHEMBL20562842 0.85 POLB (0.58) POLBHDAC6ALDH1A1ADRA1AKDM4E
SCHEMBL8196662 0.82 POLB (0.67) POLBHDAC6ALDH1A1ADRA1AHPGD
SCHEMBL16067612 0.82 POLB (0.88) POLBHDAC6ALDH1A1ADRA1AKDM4E
SCHEMBL12664048 0.82 POLB (0.67) POLBHDAC6ALDH1A1ADRA1AKDM4E
SCHEMBL10413396 0.79 POLB (0.62) POLBHDAC6ALDH1A1KDM4EHTT
SCHEMBL4580075 0.78 POLB (0.61) POLBALDH1A1KDM4EHPGDALOX15
SCHEMBL3607524 0.77 POLB (0.66) POLBHDAC6ALDH1A1KDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105452233-A Piperidine and azepane derivatives as prokineticin receptor modulators TAKEDA PHARMACEUTICALS CO 2016-03-30 CN claimed
CN-105452233-A Piperidine and azepane derivatives as prokineticin receptor modulators TAKEDA PHARMACEUTICALS CO 2016-03-30 CN disclosed