SCHEMBL28057481

SCHEMBL28057481

O=C(NCc1ccccc1)O[C@H]1Cc2ccc(F)cc2C1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BCHE P06276 9/20 0.50
NAMPT P43490 2/20 0.47
RAB9A P51151 2/20 0.46
ALDH1A1 P00352 1/20 0.46
KCNA3 P22001 1/20 0.43
PSEN1 P49768 1/20 0.43
PSEN2 P49810 1/20 0.43
APH1B Q8WW43 1/20 0.43
NCSTN Q92542 1/20 0.43
APH1A Q96BI3 1/20 0.43
PSENEN Q9NZ42 1/20 0.43
F2 P00734 1/20 0.43
PRSS1 P07477 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
POLB P06746 1/20 0.42
PLA2G1B P04054 1/20 0.42
ATG4B Q9Y4P1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27810920 0.81 BCHE (0.61) BCHERAB9AALDH1A1KCNA3F2
SCHEMBL27923505 0.80 BCHE (0.57) BCHEALDH1A1
SCHEMBL27652150 0.79 HDAC3 (0.60) BCHERAB9AALDH1A1KCNA3F2
SCHEMBL27742584 0.79 F2 (0.63) BCHERAB9AALDH1A1KCNA3F2
SCHEMBL29286125 0.78 BCHE (0.46) BCHEALDH1A1KCNA3
SCHEMBL28576382 0.78 BCHE (0.46) BCHEALDH1A1KCNA3
SCHEMBL27630590 0.77 HDAC3 (0.62) BCHERAB9AALDH1A1KCNA3F2
SCHEMBL27709635 0.76 BCHE (0.59) BCHEALDH1A1KCNA3F2PRSS1
SCHEMBL16369737 0.76 TSHR (0.59) BCHEALDH1A1
SCHEMBL27557534 0.76 MC4R (0.59) BCHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102516115-B As the antagonist of Opioid Receptors or the new compound of inverse agonist SMITHKLINE BEECHAN CORP. (US) 2016-05-11 CN disclosed