SCHEMBL28059334

SCHEMBL28059334

C=CC(=O)Nc1cccc(Nc2ncc(C(F)(F)F)c(Nc3cccc(NC(=O)C=C)c3)n2)c1

nearest known ligand 0.85

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BTK Q06187 10/20 0.85
EGFR P00533 11/20 0.83
JAK3 P52333 5/20 0.83
JAK2 O60674 3/20 0.83
ITK Q08881 2/20 0.69
ERBB2 P04626 1/20 0.67
ERBB3 P21860 1/20 0.67
ERBB4 Q15303 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29722371 0.97 BTK (0.82) BTKEGFRJAK3JAK2ITK
SCHEMBL12519708 0.97 BTK (0.82) BTKEGFRJAK3JAK2ITK
SCHEMBL12519518 0.91 EGFR (1.00) BTKEGFRJAK3JAK2ITK
SCHEMBL29722500 0.91 EGFR (1.00) BTKEGFRJAK3JAK2ITK
SCHEMBL18970349 0.90 EGFR (0.72) BTKEGFRJAK3JAK2ERBB2
SCHEMBL12519713 0.89 EGFR (0.77) BTKEGFRJAK3JAK2ITK
SCHEMBL24900775 0.89 BTK (0.69) BTKEGFRJAK3JAK2ITK
SCHEMBL9924738 0.89 BTK (0.69) BTKEGFRJAK3JAK2ERBB2
SCHEMBL17197240 0.89 BTK (0.69) BTKEGFRJAK3JAK2ERBB2
SCHEMBL12519783 0.89 EGFR (0.85) BTKEGFRJAK3JAK2ITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384695-A Pyrimidine derivative, preparation method therefor and application thereof in medicine SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-03-09 CN disclosed